Unlocking Undruggable Targets: Shifting Paradigms in Modern Drug Discovery
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Pharmacokinetics
Also known as:
Pharmacokinetic
Drug Trials
Drug
Drug Name
Drug Description
Drug
Drug Name
Target
Type
Drug
Drug Name
Phase
Status
Count
DB05812
Abiraterone
0
Active Not Recruiting
1
DB00594
Amiloride
0
Completed
1
DB14726
Dabigatran
0
Completed
1
DB00080
Daptomycin
0
Completed
1
DB01167
Itraconazole
0
Completed
1
DB15257
Milademetan
0
Completed
1
DB01263
Posaconazole
0
Completed
1
DB12874
Quizartinib
0
Completed
1
DB01045
Rifampicin
0
Completed
1
DB14010
5-methoxy-N,N-dimethyltryptamine
1
Completed
1
DB15333
AZD-1386
1
Completed
1
DB12576
AZD-3043
1
Withdrawn
1
DB16822
AZD-5069
1
Completed
1
DB11804
AZD-5672
1
Completed
2
DB13994
AZD-7325
1
Suspended
1
DB15418
AZD-9977
1
Completed
1
DB15418
AZD-9977
1
Withdrawn
1
DB05812
Abiraterone
1
Completed
1
DB11703
Acalabrutinib
1
Completed
1
DB00316
Acetaminophen
1
Completed
1
DB00819
Acetazolamide
1
Completed
1
DB00945
Acetylsalicylic acid
1
Completed
3
DB00051
Adalimumab
1
Completed
1
DB09302
Alirocumab
1
Completed
1
DB06673
Almorexant
1
Completed
1
DB00404
Alprazolam
1
Completed
1
DB11863
Alvelestat
1
Withdrawn
1
DB00613
Amodiaquine
1
Recruiting
1
DB01060
Amoxicillin
1
Completed
1
DB01217
Anastrozole
1
Completed
1
DB11976
Anifrolumab
1
Completed
1
DB06605
Apixaban
1
Completed
1
DB05676
Apremilast
1
Completed
1
DB06697
Artemether
1
Recruiting
1
DB00126
Ascorbic acid
1
Completed
2
DB01076
Atorvastatin
1
Completed
2
DB00572
Atropine
1
Recruiting
1
DB09060
Avibactam
1
Completed
1
DB00207
Azithromycin
1
Completed
1
DB00207
Azithromycin
1
Unknown Status
1
DB00181
Baclofen
1
Completed
1
DB12299
Bavisant
1
Completed
2
DB12299
Bavisant
1
Withdrawn
1
DB00394
Beclomethasone dipropionate
1
Completed
1
DB00112
Bevacizumab
1
Completed
1
DB00112
Bevacizumab
1
Withdrawn
1
DB11591
Bilastine
1
Unknown Status
1
DB17452
Boserolimab
1
Active Not Recruiting
1
DB09019
Bromhexine
1
Not Yet Recruiting
1
DB01222
Budesonide
1
Completed
1
DB00921
Buprenorphine
1
Completed
1
DB00201
Caffeine
1
Completed
1
DB09061
Cannabidiol
1
Completed
1
DB09061
Cannabidiol
1
Recruiting
1
DB12218
Capivasertib
1
Active Not Recruiting
1
DB12218
Capivasertib
1
Completed
1
DB00190
Carbidopa
1
Completed
1
DB00958
Carboplatin
1
Active Not Recruiting
1
DB12830
Cebranopadol
1
Completed
2
DB01327
Cefazolin
1
Recruiting
1
DB01413
Cefepime
1
Completed
1
DB14879
Cefiderocol
1
Active Not Recruiting
1
DB01415
Ceftibuten
1
Completed
2
DB00482
Celecoxib
1
Completed
2
DB00608
Chloroquine
1
Completed
1
DB00356
Chlorzoxazone
1
Completed
2
DB00537
Ciprofloxacin
1
Completed
2
DB04272
Citric acid
1
Completed
1
DB01211
Clarithromycin
1
Completed
5
DB00882
Clomifene
1
Completed
2
DB01068
Clonazepam
1
Completed
1
DB00758
Clopidogrel
1
Completed
1
DB09065
Cobicistat
1
Completed
1
DB00907
Cocaine
1
Completed
1
DB01394
Colchicine
1
Completed
12
DB00091
Cyclosporine
1
Completed
2
DB11908
Dapivirine
1
Completed
1
DB12289
Darexaban
1
Completed
2
DB12941
Darolutamide
1
Completed
2
DB01264
Darunavir
1
Completed
1
DB01254
Dasatinib
1
Completed
1
DB06444
Dexanabinol
1
Completed
1
DB11807
Dexmecamylamine
1
Completed
1
DB00633
Dexmedetomidine
1
Completed
1
DB00586
Diclofenac
1
Completed
1
DB00390
Digoxin
1
Completed
2
DB00343
Diltiazem
1
Completed
3
DB00204
Dofetilide
1
Completed
2
DB00470
Dronabinol
1
Completed
1
DB00470
Dronabinol
1
Recruiting
1
DB00625
Efavirenz
1
Completed
4
DB15001
Eflapegrastim
1
Completed
1
DB05187
Elafibranor
1
Completed
2
DB09038
Empagliflozin
1
Completed
1
DB06735
Enclomiphene
1
Completed
1
DB06423
Endostatin
1
Completed
1
DB00494
Entacapone
1
Completed
1
DB05094
Enzalutamide
1
Completed
1
DB08899
Enzalutamide
1
Completed
1
DB00700
Eplerenone
1
Withdrawn
1
DB00199
Erythromycin
1
Completed
1
DB00736
Esomeprazole
1
Completed
3
DB00736
Esomeprazole
1
Unknown Status
1
DB00783
Estradiol
1
Completed
1
DB00977
Ethinylestradiol
1
Completed
6
DB00977
Ethinylestradiol
1
Suspended
1
DB06414
Etravirine
1
Completed
1
DB01590
Everolimus
1
Completed
1
DB09303
Evolocumab
1
Completed
1
DB00973
Ezetimibe
1
Completed
4
DB13873
Fenofibric acid
1
Completed
2
DB00950
Fexofenadine
1
Completed
1
DB16165
Finerenone
1
Completed
2
DB12030
Fluorescein lisicol
1
Completed
1
DB06623
Flupirtine
1
Completed
1
DB00158
Folic acid
1
Completed
5
DB00066
Follitropin
1
Completed
1
DB12010
Fostamatinib
1
Completed
4
DB14041
Fremanezumab
1
Completed
1
DB00947
Fulvestrant
1
Active Not Recruiting
1
DB00947
Fulvestrant
1
Completed
1
DB11769
Funapide
1
Completed
1
DB17499
GB1211
1
Completed
1
DB08872
Gabapentin enacarbil
1
Completed
1
DB17084
Gadopiclenol
1
Completed
1
DB00674
Galantamine
1
Completed
1
DB01241
Gemfibrozil
1
Completed
1
DB00222
Glimepiride
1
Completed
1
DB00889
Granisetron
1
Completed
1
DB06261
Hexaminolevulinate
1
Completed
1
DB12101
Iberdomide
1
Completed
1
DB12471
Ibrexafungerp
1
Completed
2
DB01050
Ibuprofen
1
Completed
1
DB11964
Ilaprazole
1
Completed
1
DB11964
Ilaprazole
1
Not Yet Recruiting
1
DB11964
Ilaprazole
1
Recruiting
1
DB12105
Imagabalin
1
Completed
1
DB12105
Imagabalin
1
Terminated
1
DB00060
Interferon beta-1a
1
Completed
1
DB05382
Iodine
1
Completed
1
DB01020
Isosorbide mononitrate
1
Withdrawn
1
DB01167
Itraconazole
1
Completed
6
DB01167
Itraconazole
1
Not Yet Recruiting
1
DB01167
Itraconazole
1
Recruiting
1
DB15173
JNJ-42165279
1
Completed
1
DB01322
Kava
1
Completed
1
DB01221
Ketamine
1
Unknown Status
1
DB01026
Ketoconazole
1
Completed
6
DB00465
Ketorolac
1
Completed
1
DB16956
L-Acetylleucine
1
Not Yet Recruiting
1
DB16956
L-Acetylleucine
1
Recruiting
1
DB16956
L-Acetylleucine
1
Unknown Status
1
DB14801
Lanifibranor
1
Completed
1
DB06685
Laquinimod
1
Completed
1
DB01235
Levodopa
1
Completed
1
DB00367
Levonorgestrel
1
Completed
2
DB00451
Levothyroxine
1
Completed
2
DB00281
Lidocaine
1
Completed
1
DB13200
Lipegfilgrastim
1
Completed
1
DB18054
Lisaftoclax
1
Completed
1
DB01601
Lopinavir
1
Completed
1
DB00678
Losartan
1
Completed
1
DB14596
Loteprednol etabonate
1
Completed
1
DB06708
Lumefantrine
1
Recruiting
1
DB08815
Lurasidone
1
Completed
2
DB15028
MK-1064
1
Completed
1
DB00742
Mannitol
1
Completed
1
DB00351
Megestrol acetate
1
Completed
1
DB01065
Melatonin
1
Completed
1
DB00814
Meloxicam
1
Completed
1
DB06612
Mepolizumab
1
Completed
1
DB00331
Metformin
1
Completed
4
DB00331
Metformin
1
Unknown Status
1
DB00422
Methylphenidate
1
Completed
1
DB00264
Metoprolol
1
Completed
1
DB00379
Mexiletine
1
Completed
1
DB14158
Microcrystalline cellulose
1
Completed
2
DB00683
Midazolam
1
Completed
2
DB01454
Midomafetamine
1
Completed
1
DB01454
Midomafetamine
1
Not Yet Recruiting
1
DB01017
Minocycline
1
Completed
1
DB08893
Mirabegron
1
Completed
6
DB00218
Moxifloxacin
1
Completed
7
DB14011
Nabiximols
1
Recruiting
1
DB12598
Nafamostat
1
Completed
2
DB00844
Nalbuphine
1
Terminated
1
DB06230
Nalmefene
1
Completed
1
DB01183
Naloxone
1
Completed
1
DB00704
Naltrexone
1
Completed
1
DB06682
Naproxcinod
1
Completed
1
DB00788
Naproxen
1
Completed
3
DB00627
Niacin
1
Recruiting
1
DB00699
Nicergoline
1
Completed
1
DB02701
Nicotinamide
1
Completed
1
DB16691
Nirmatrelvir
1
Completed
1
DB14678
Norethindrone enanthate
1
Completed
1
DB00717
Norethisterone
1
Completed
1
DB00957
Norgestimate
1
Completed
5
DB00957
Norgestimate
1
Suspended
1
DB00334
Olanzapine
1
Completed
1
DB13127
Olokizumab
1
Completed
1
DB09568
Omega-3-carboxylic acids
1
Completed
1
DB00338
Omeprazole
1
Completed
3
DB00497
Oxycodone
1
Completed
1
DB01229
Paclitaxel
1
Active Not Recruiting
1
DB14977
Padsevonil
1
Completed
1
DB00213
Pantoprazole
1
Completed
1
DB00019
Pegfilgrastim
1
Unknown Status
1
DB09122
Peginterferon beta-1a
1
Completed
1
DB09037
Pembrolizumab
1
Active Not Recruiting
1
DB00642
Pemetrexed
1
Active Not Recruiting
1
DB00252
Phenytoin
1
Recruiting
1
DB01100
Pimozide
1
Completed
1
DB01132
Pioglitazone
1
Completed
1
DB09287
Polyethylene glycol
1
Completed
1
DB12016
Ponesimod
1
Completed
1
DB00761
Potassium chloride
1
Completed
1
DB01708
Prasterone
1
Completed
1
DB00860
Prednisolone
1
Completed
1
DB01087
Primaquine
1
Withdrawn
1
DB00396
Progesterone
1
Completed
4
DB11664
Psilocybin
1
Completed
1
DB00468
Quinine
1
Completed
2
DB12874
Quizartinib
1
Completed
1
DB01129
Rabeprazole
1
Completed
2
DB08913
Radium Ra 223 dichloride
1
Completed
1
DB06817
Raltegravir
1
Completed
1
DB00863
Ranitidine
1
Completed
3
DB00243
Ranolazine
1
Completed
1
DB08896
Regorafenib
1
Completed
2
DB06602
Reslizumab
1
Completed
1
DB02709
Resveratrol
1
Completed
1
DB01045
Rifampicin
1
Completed
2
DB01220
Rifaximin
1
Completed
1
DB05083
Rilpivirine
1
Completed
1
DB08864
Rilpivirine
1
Completed
1
DB14924
Ritlecitinib
1
Completed
1
DB00503
Ritonavir
1
Completed
3
DB06228
Rivaroxaban
1
Completed
2
DB15078
Rogaratinib
1
Completed
1
DB05332
Romiplostim
1
Recruiting
1
DB01098
Rosuvastatin
1
Completed
3
DB01098
Rosuvastatin
1
Recruiting
1
DB11362
Selexipag
1
Completed
1
DB06290
Simeprevir
1
Completed
1
DB00641
Simvastatin
1
Recruiting
1
DB00877
Sirolimus
1
Completed
1
DB14482
Sodium ascorbate
1
Completed
1
DB01390
Sodium bicarbonate
1
Completed
1
DB09153
Sodium chloride
1
Completed
2
DB09472
Sodium sulfate
1
Completed
1
DB01591
Solifenacin
1
Completed
6
DB00398
Sorafenib
1
Completed
1
DB00708
Sufentanil
1
Completed
2
DB00795
Sulfasalazine
1
Completed
1
DB00864
Tacrolimus
1
Completed
2
DB00706
Tamsulosin
1
Completed
4
DB16338
Taniborbactam
1
Completed
1
DB06204
Tapentadol
1
Completed
4
DB16690
Tegoprazan
1
Completed
1
DB16690
Tegoprazan
1
Unknown Status
1
DB05253
Telapristone acetate
1
Completed
1
DB00624
Testosterone
1
Completed
1
DB00277
Theophylline
1
Completed
2
DB04902
Ticagrelor
1
Completed
1
DB08816
Ticagrelor
1
Completed
2
DB08816
Ticagrelor
1
Recruiting
1
DB06273
Tocilizumab
1
Completed
1
DB00193
Tramadol
1
Completed
3
DB00656
Trazodone
1
Completed
1
DB00209
Trospium
1
Completed
1
DB12099
UK-396,082
1
Completed
1
DB12255
Vadadustat
1
Completed
1
DB00177
Valsartan
1
Completed
1
DB01273
Varenicline
1
Completed
2
DB16347
Velsecorat
1
Completed
1
DB00661
Verapamil
1
Completed
2
DB15456
Vericiguat
1
Completed
1
DB05700
Vortioxetine
1
Completed
1
DB15154
Vunakizumab
1
Unknown Status
1
DB00682
Warfarin
1
Completed
1
DB00682
Warfarin
1
Withdrawn
1
DB00613
Amodiaquine
1 / 2
Terminated
1
DB06697
Artemether
1 / 2
Terminated
1
DB09050
Ceftolozane
1 / 2
Completed
1
DB08884
Gadoxetic acid
1 / 2
Completed
1
DB06708
Lumefantrine
1 / 2
Terminated
1
DB01087
Primaquine
1 / 2
Terminated
1
DB00203
Sildenafil
1 / 2
Completed
1
DB01606
Tazobactam
1 / 2
Completed
1
DB09299
Tenofovir alafenamide
1 / 2
Recruiting
1
DB00207
Azithromycin
2
Completed
1
DB11808
Faldaprevir
2
Completed
1
DB08906
Fluticasone furoate
2
Completed
1
DB01322
Kava
2
Completed
1
DB00218
Moxifloxacin
2
Completed
1
DB11816
Omecamtiv Mecarbil
2
Completed
1
DB00811
Ribavirin
2
Completed
1
DB09082
Vilanterol
2
Completed
1
DB00582
Voriconazole
2
Completed
1
DB18673
XEN-D0501
2
Completed
1
DB00051
Adalimumab
2 / 3
Recruiting
1
DB00633
Dexmedetomidine
2 / 3
Completed
1
DB15341
Dinalbuphine sebacate
2 / 3
Recruiting
1
DB01306
Insulin aspart
2 / 3
Completed
1
DB00030
Insulin human
2 / 3
Completed
1
DB11206
Bemotrizinol
3
Completed
1
DB09038
Empagliflozin
3
Completed
1
DB09496
Octinoxate
3
Completed
1
DB00864
Tacrolimus
3
Completed
1
DB01001
Albuterol
4
Completed
1
DB01060
Amoxicillin
4
Recruiting
1
DB06605
Apixaban
4
Completed
1
DB01238
Aripiprazole
4
Completed
1
DB01117
Atovaquone
4
Withdrawn
1
DB00207
Azithromycin
4
Recruiting
1
DB00297
Bupivacaine
4
Recruiting
1
DB09050
Ceftolozane
4
Terminated
1
DB01394
Colchicine
4
Completed
1
DB06700
Desvenlafaxine
4
Completed
2
DB01234
Dexamethasone
4
Active Not Recruiting
1
DB00633
Dexmedetomidine
4
Completed
1
DB00633
Dexmedetomidine
4
Unknown Status
1
DB00668
Epinephrine
4
Completed
1
DB00056
Gemtuzumab ozogamicin
4
Completed
1
DB01167
Itraconazole
4
Completed
1
DB00130
L-Glutamine
4
Completed
1
DB09415
Meglumine
4
Completed
1
DB00916
Metronidazole
4
Recruiting
1
DB00683
Midazolam
4
Completed
1
DB00497
Oxycodone
4
Active Not Recruiting
1
DB01263
Posaconazole
4
Recruiting
1
DB01131
Proguanil
4
Withdrawn
1
DB12404
Remimazolam
4
Active Not Recruiting
1
DB06206
Sugammadex
4
Recruiting
2
DB06206
Sugammadex
4
Unknown Status
1
DB01015
Sulfamethoxazole
4
Completed
1
DB00864
Tacrolimus
4
Completed
1
DB00675
Tamoxifen
4
Completed
1
DB01606
Tazobactam
4
Terminated
1
DB00208
Ticlopidine
4
Completed
1
DB00440
Trimethoprim
4
Completed
1
DB00209
Trospium
4
Completed
1
DB00313
Valproic acid
4
Terminated
1
DB00316
Acetaminophen
Not Available
Completed
1
DB00316
Acetaminophen
Not Available
Withdrawn
1
DB00381
Amlodipine
Not Available
Withdrawn
1
DB01060
Amoxicillin
Not Available
Completed
1
DB01053
Benzylpenicillin
Not Available
Active Not Recruiting
1
DB01053
Benzylpenicillin
Not Available
Completed
1
DB00297
Bupivacaine
Not Available
Completed
1
DB00201
Caffeine
Not Available
Completed
1
DB00520
Caspofungin
Not Available
Recruiting
1
DB01212
Ceftriaxone
Not Available
Recruiting
1
DB00567
Cephalexin
Not Available
Completed
1
DB00215
Citalopram
Not Available
Completed
1
DB00766
Clavulanic acid
Not Available
Completed
1
DB00879
Emtricitabine
Not Available
Completed
1
DB01175
Escitalopram
Not Available
Completed
2
DB00736
Esomeprazole
Not Available
Completed
1
DB00977
Ethinylestradiol
Not Available
Completed
1
DB00294
Etonogestrel
Not Available
Completed
1
DB00196
Fluconazole
Not Available
Recruiting
1
DB01067
Glipizide
Not Available
Completed
1
DB01050
Ibuprofen
Not Available
Completed
1
DB00030
Insulin human
Not Available
Completed
1
DB09332
Kappadione
Not Available
Completed
1
DB01221
Ketamine
Not Available
Completed
1
DB01221
Ketamine
Not Available
Not Yet Recruiting
1
DB06218
Lacosamide
Not Available
Completed
1
DB01202
Levetiracetam
Not Available
Completed
1
DB00760
Meropenem
Not Available
Completed
1
DB00760
Meropenem
Not Available
Recruiting
1
DB00264
Metoprolol
Not Available
Completed
1
DB00683
Midazolam
Not Available
Completed
2
DB00370
Mirtazapine
Not Available
Completed
1
DB15661
Molnupiravir
Not Available
Completed
1
DB18740
Nogapendekin alfa
Not Available
Terminated
1
DB01174
Phenobarbital
Not Available
Completed
1
DB00252
Phenytoin
Not Available
Completed
1
DB01022
Phylloquinone
Not Available
Completed
1
DB00863
Ranitidine
Not Available
Completed
1
DB01104
Sertraline
Not Available
Completed
1
DB00864
Tacrolimus
Not Available
Unknown Status
1
DB12343
Temocillin
Not Available
Recruiting
2
DB00300
Tenofovir disoproxil
Not Available
Completed
1
DB01610
Valganciclovir
Not Available
Completed
1
DB00313
Valproic acid
Not Available
Completed
1
DB00512
Vancomycin
Not Available
Not Yet Recruiting
1
DB00285
Venlafaxine
Not Available
Completed
1
DB00682
Warfarin
Not Available
Completed
1