Cytochrome P-450 CYP2C9 Inducers (moderate)

Name
Cytochrome P-450 CYP2C9 Inducers (moderate)
Accession Number
DBCAT003109
Description

Not Available

Drugs
DrugDrug Description
BosentanA dual endothelin receptor antagonist used to treat pulmonary arterial hypertension.
EnzalutamideA second-generation androgen receptor inhibitor used to treat castration-resistant prostate cancer and metastatic castration-sensitive prostate cancer.
AlpelisibAlpelisib is indicated in combination with fulvestrant to treat postmenopausal women, and men, with advanced or metastatic breast cancer. This cancer must be hormone receptor (HR)-positive, human epidermal growth factor...
RifampinAn antibiotic used alone or in combination with other antimicrobial drugs to treat tuberculosis and asymptomatic carriers of Neisseria meningitidis.
Drugs & Drug Targets
DrugTargetType
BosentanEndothelin B receptortarget
BosentanEndothelin-1 receptortarget
BosentanCytochrome P450 3A4enzyme
BosentanCytochrome P450 2C9enzyme
BosentanBile salt export pumptransporter
EnzalutamideSerum albumincarrier
EnzalutamideCytochrome P450 2C8enzyme
EnzalutamideCytochrome P450 3A4enzyme
EnzalutamideAndrogen receptortarget
EnzalutamideCytochrome P450 2C9enzyme
EnzalutamideCytochrome P450 2C19enzyme
EnzalutamideCytochrome P450 2B6enzyme
EnzalutamideCytochrome P450 3A5enzyme
EnzalutamideP-glycoprotein 1transporter
AlpelisibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformtarget
AlpelisibCytochrome P450 3A4enzyme
AlpelisibCytochrome P450 2C9enzyme
AlpelisibCytochrome P450 2C8enzyme
AlpelisibCytochrome P450 2C19enzyme
AlpelisibATP-binding cassette sub-family G member 2transporter
AlpelisibP-glycoprotein 1transporter
RifampinNuclear receptor subfamily 1 group I member 2target
RifampinCytochrome P450 3A4enzyme
RifampinCytochrome P450 1A2enzyme
RifampinCytochrome P450 2C8enzyme
RifampinUDP-glucuronosyltransferase 1-1enzyme
RifampinCytochrome P450 2C9enzyme
RifampinCytochrome P450 2B6enzyme
RifampinCytochrome P450 2C19enzyme
RifampinCanalicular multispecific organic anion transporter 2transporter
RifampinMultidrug resistance-associated protein 5transporter
RifampinP-glycoprotein 1transporter
RifampinCanalicular multispecific organic anion transporter 1transporter
RifampinSolute carrier organic anion transporter family member 2B1transporter
RifampinBile salt export pumptransporter
RifampinMultidrug resistance-associated protein 1transporter
RifampinSolute carrier organic anion transporter family member 1A2transporter
RifampinSolute carrier organic anion transporter family member 1B3transporter
RifampinSolute carrier family 22 member 7transporter
RifampinSolute carrier organic anion transporter family member 1B1transporter
RifampinCytochrome P450 2A6enzyme
RifampinCytochrome P450 2E1enzyme
RifampinCytochrome P450 3A43enzyme
RifampinCytochrome P450 3A7enzyme
RifampinSolute carrier family 22 member 6transporter
RifampinSolute carrier family 22 member 8transporter
RifampinUDP-glucuronosyltransferase 1-9enzyme
RifampinCytochrome P450 3A5enzyme
RifampinSerum albumincarrier
Rifampinalpha1-acid glycoproteincarrier
RifampinDNA-directed RNA polymerase subunit betatarget